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乐贵洲

2019-12-07     (浏览次数:)     打印    收藏

 

乐贵洲   

职称:副教授   

所属系室应用化学系

导师类别:硕士生导师     最高学位:理学博士

Tel:0835-2886189  Email :yueguizhou@sicau.edu.cn;14640775@qq.com

 < 个人简历 >

毕业学校四川大学

招收硕士专业:生物资源化学(学硕);生物与医药(专硕)   

招收方向:

1.有机方法学

2.活性有机小分子的设计、合成及开发

已指导硕士人数:7人

主要讲授课程有机化学、有机合成、绿色化学及药物合成等

主要学习和工作经历:

19989-20026月     湖北民族学院 本科

20029-20056月     湖北大学    硕士研究生

20057-200812月   美高梅MGM33999 助教

20089-201112月   四川大学     博士研究生

20091-201212月   美高梅MGM33999 讲师

20131-至今                美高梅MGM33999 副教授

20143-20152月     新加坡南洋理工大学 访问学者

< 主要学术论文 >

1.Guizhou Yue, Kaining Lei, Hajime Hirao, Jianrong (Steve) Zhou* Palladium-Catalyzed Asymmetric Reductive Heck Reaction of Aryl Halides. Angewandte Chemie International Edition 2015, 54, 6531-6535.(一区, TOP

2.Guizhou Yue, Li Yang, Changchun Yuan, Xiaoling Jiang, Bo Liu*. Total Synthesis of (±)-Chloranthalactone A. Organic Letters 2011, 13, 5406-5408.(一区)

3.Guizhou Yue*Dan JiangZhengjie Dou, Sicheng Li, Juhua Feng, Li Zhang, Huabao Chen, Chunping Yang, Zhongqiong Yin, Xu Song, Xiaoxia Liang, Xianxiang Wang, Cuifen Lu. Rapid umpolung Michael addition of isatin N,N′-cyclic azomethine imine 1,3-dipoles with chalcones. New Journal of Chemistry 2021, 45, 11712-11718.(三区)

4.Guizhou Yue*, Dou Z., Zhou Z., Zhang L., Feng J., Chen H., Yin Z., Song X., Liang X., Wang X., Rao H., Lu C. Rapid abnormal [3+2]-cycloaddition of isatin N,N′-cyclic azomethine imine 1,3-dipoles with chalcones. New Journal of Chemistry 2020, 44, 8813-8817.(三区)

5.Guizhou Yue*, Wu Y., Dou Z., Chen H., Yin Z., Song X., He C., Wang X., Feng J., Zhang Z., Zou P., Lu C. Synthesis of Spiropyrrolidine Oxindoles via Ag-catalyzed Stereo- and Regioselective 1,3-diploar Cycloaddition of Indole-based Azomethine Ylides with Chalcones. New Journal of Chemistry 2018, 42, 20024-20031.(三区)

6.Guizhou Yue*, Li S., Jiang D., Ding G., Feng J., Chen H., Yang C., Yin Z., Song X., Liang X., Zhang L., Wang X., Lu C. Syntheses of 3,3-Disubstituted Dihydrobenzofurans, Indolines, Indolinones and Isochromanes by Palladium-Catalyzed Tandem Reaction Using Pd(PPh3)2Cl2/(±)-BINAP as a Catalytic System. Catalysts 2020, 10, 1084.(三区)

7.Guizhou Yue*, Wu Y., Wu C., Yin Z., Chen H., Wang X., Zhang Z. Synthesis of 2-arylindoles by Suzuki coupling reaction of 3-bromoindoles with hindered benzoboronic acids. Tetrahedron Lett. 2017, 58, 666-669.(三区)

8.Guizhou Yue, Li Yang, Changchun Yuan, Biao Du, and Bo Liu*. Total Syntheses of Lindenane-type Sesquiterpenoids: (±)-Chloranthalactones A, B, F, (±)-9-Hydroxy Heterogorgiolide, and (±)-Shizukanolide E. Tetrahedron 2012, 68, 9624-9637.(三区)

9.Guizhou Yue, Yadong Wan, Shaojun Song, Guichun Yang, Zuxing Chen*. Synthesis of a Library of Benzoindolizines using Poly(ethylene glycol) as Soluble Support. Bioorganic & Medicinal Chemistry Letters 2005, 15, 453-458.(三区)

10.Guizhou Yue*, Zuxing Chen, Guichun Yang. Synthesis of a Library of 1,2,3,7-Tetrasubstituted Indolizines using Poly(ethylene glycol) as Soluble Support. Journal of Heterocyclic Chemistry 2006, 43, 781-786. (四区)

11.乐贵洲*, 刘波*. 1,3-偶极子[3+n](n≥3)环加成反应的研究进展. 有机化学, 2020, 40, 3132-3153.(三区)

12.乐贵洲, 黄轩, 刘波*. 具有反式六氢茚满结构的萜类化合物的合成研究进展. 有机化学2013, 33, 1167-1185.(三区)

13.乐贵洲, 杨立, 袁长春, 杜彪, 刘波*. 乌药烷型倍半萜及其二聚体的全合成研究进展. 有机化学 2012, 33, 90-100.(三区)

14.乐贵洲*, 黄乾明, 邹平. 倍半萜englerin A及其类似物的合成. 化学进展2012, 24, 1742-1750.(四区)

15.乐贵洲*, 黄乾明, 邹平. 中氮茚的合成研究进展. 有机化学 2007, 27, 1060-1068.(三区)

16.Guizhou Yue*, Kai Meng, Qin Liu. One‐Step Synthesis of N‐Doped Carbon and Its Application as a Cost‐Efficient Catalyst for the Oxygen Reduction Reaction in Microbial Fuel Cells. ChemPlusChem 2015, 80, 1133-1138.(三区)

17.Guizhou Yue, Suying Li, Wei Liu, Fang Ding, Ping Zou, Xianxiang Wang, Qingbiao Zhao, Hanbing Rao*. Ratiometric fluorescence based on silver clusters and N, Fe doped carbon dots for determination of H2O2 and UA: N, Fe doped carbon dots as mimetic peroxidaseSensors and Actuators B: Chemical2019, 287, 408-415.(一区)

18.Chunlin Wu, Guizhou Yue, Christian Duc-Trieu Nielsen, Kai Xu, Hajime Hirao, Jianrong (Steve) Zhou.* Asymmetric Conjugate Addition of Organoboron Reagents to Common Enones Using Copper Catalysts. Journal of the American Chemical Society 2016, 138, 742-745.(一区, TOP

19.Yinjun, Zou, Guizhou Yue, Jianwei Xu, Jianrong Zhou Steve.* General Suzuki Coupling of Heteroaryl Bromides by Using Tri‐tert‐butylphosphine as a Supporting Ligand. European Journal of Organic Chemistry 2014, 27, 5901-5905.

20.Li Yang, Guizhou Yue, Changchun Yuan, Bo Liu.* Synthetic Studies toward Lindenane-Type Sesquiterpenoid Dimers. Synlett 2014, 25, 2471-2474.(三区)

21.Zuxing Chen*, Guizhou Yue, Cuifen Lu, Guichun Yang. Synthesis of a Library of Indolizines using Poly(ethylene glycol) as Soluble Support. Synlett 2004, 1231-1234.(三区)

22.Xiaojin Wu, Chuanhu Lei, Guizhou Yue, Jianrong Zhou Steve.* Palladium‐Catalyzed Direct Cyclopropylation of Heterocycles. Angewandte Chemie International Edition 2015, 54, 9601-9605.(一区, TOP

23.Changchun Yuan, Li Yang, Guizhou Yue, Tianzi Yu, Weiming Zhong and Bo Liu.* A Base-Promoted Deprotection of 1,3-Dioxolanes to Ketones. Tetrahedron Letters 2012, 53, 6972-6976.(三区)

24.吴瑶, 豆正杰, 陈华保, 乐贵洲*. 2,4,6-三甲基苯硼酸及其酯在偶联反应中的应用. 有机化学, 2018, 38, 2896-2926.(三区)

25.丁刚, 王泽宇, 殷中琼, 乐贵洲*. 钯催化的串联反应构建苯并五元杂环的研究进展. 有机化学 2016, 36, 53-59.(三区)

26.何桥, 殷中琼, 陈华保, 张祖民, 王显祥, 乐贵洲*. 茚及其衍生物的催化不对称合成. 化学进展 2016, 28, 801-813.(四区)

< 授权发明专利/软件著作权 >

1.乐贵洲、何桥、吴瑶、张祖民,“一种苯并吡喃酮类化合物及其制备方法和应用”,专利证号:ZL201810550598.X,授权公告号:CN 108822065 B

< 科研项目及成果获奖(含专利、新品种) >

1. 伪狂犬病毒小分子抑制剂的合成、构效关系研究与应用,四川省科技厅国际合作研究项目(2020YFH0129),20万元,2020-2022年,在研,主持。

2. 可溶性聚合物支载组合合成具有生物活性的含氮杂环化合物,四川省科技厅应用基础研究项目(2012JY0118),10万元,2012-2016年,结题,主持;

3、倍半萜onoseriolide的全合成研究,四川省教育厅科研项目(11AZ071),3万元,2011-2014年,结题,主持。